Cathepsin Inhibitor 1

CAS No. 225120-65-0

Cathepsin Inhibitor 1( Cathepsin Inhibitor 1 | Cathepsin-Inhibitor-1 | CTS-IN-1 )

Catalog No. M18263 CAS No. 225120-65-0

Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 87 Get Quote
10MG 140 Get Quote
25MG 267 Get Quote
50MG 507 Get Quote
100MG 731 Get Quote
500MG 1503 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Cathepsin Inhibitor 1
  • Note
    Research use only, not for human use.
  • Brief Description
    Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively.
  • Description
    Cathepsin Inhibitor 1 is a pan-inhibitor of Cathepsin (L, L2, S, K, B).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Cathepsin Inhibitor 1 | Cathepsin-Inhibitor-1 | CTS-IN-1
  • Pathway
    Immunology/Inflammation
  • Target
    Antiviral
  • Recptor
    Cathepsin K| Cathepsin L| Cathepsin L2| Cathepsin S| Cathepsin S
  • Research Area
    Others-Field
  • Indication
    ——

Chemical Information

  • CAS Number
    225120-65-0
  • Formula Weight
    401.89
  • Molecular Formula
    C20H24ClN5O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (248.82 mM)
  • SMILES
    CN1N=C(C=C1C(=O)N[C@@H](CC1=CC=CC(Cl)=C1)C(=O)NCC#N)C(C)(C)C
  • Chemical Name
    (S)-3-(tert-butyl)-N-(3-(3-chlorophenyl)-1-((cyanomethyl)amino)-1-oxopropan-2-yl)-1-methyl-1H-pyrazole-5-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Asaad N, et al. Bioorg Med Chem Lett, 2009, 19(15), 4280-4283.
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